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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T0218 | Biperiden | Bipariden,Akineton,KL 373,Biperidine | AChR |
Biperiden (Bipariden) is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, idiopathic, and postencephalitic parkinsonism. ... | |||
T9771 | Velufenacin | AChR | |
Velufenacin is an antagonist of muscarinic receptor[1]. | |||
T23297 | (S)-(+)-Dimethindene maleate | AChR , Histamine Receptor | |
(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1, M3, and M4 receptors. | |||
T16989 | Tarafenacin D-tartrate | SVT-40776 D-tartrate | Others |
Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor. | |||
T13992 | CHF5407 | SVT-47060 | AChR |
CHF5407(SVT-47060) is a potent and selective muscarinic M3 receptor antagonist with prolonged action at muscarinic receptors.CHF5407 has an effect on bronchospasm and may be used in the study of respiratory disorders.CHF... | |||
T13385 | Zamifenacin fumarate | UK-76654 fumarate | AChR |
Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor. | |||
T6364 | Desfesoterodine | 5-HMT,(R)-5-Hydroxymethyl Tolterodine,PNU-200577,5-HM,5-hydroxymethyl Tolterodine | AChR |
Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM. | |||
T7895 | Syn-Ake acetate | Dipeptide diaminobutyroyl benzylamide | AChR |
Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist. | |||
T10914L | Cyclodrine | Cyclopent | AChR |
Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist. | |||
T10914 | Cyclodrine hydrochloride | AChR | |
Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of neurologically related diseases. | |||
T1542 | Pirenzepine dihydrochloride | Pirenzepine HCl,Bisvanil,Tabe,LS519 | AChR |
Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion. | |||
T31207 | GSK233705 | Darotropium bromide,GSK 233705,GSK-233705B,GSK233705,GSK233705B,GSK-233705,GSK 233705B | AChR |
GSK233705 (Darotropium bromide) is a muscarinic receptor antagonist used in conjunction with the prevention and treatment of chronic obstructive pulmonary disease (COPD) and asthma in humans. | |||
T5655 | MAChR-IN-1 hydrochloride | AChR | |
mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm. | |||
T23508 | VU 0255035 | AChR | |
muscarinic M1 antagonist | |||
T29687 | Afacifenacin | Afacifenacin fumarate,SMP-986,NS 986,NS-986,SMP 986,NS986,SMP986 | AChR |
Afacifenacin (SMP-986) fumarate is an M3 muscarinic receptor-selective antagonist used in the study of ischemic heart disease, urinary incontinence and cystitis and other disorders. | |||
T1534 | Darifenacin hydrobromide | Darifenacin HBr,UK-88525 | AChR |
Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and overactive bladder syndrome. | |||
T28722 | SCH 57790 | SCH57790,SCH-57790 | AChR |
SCH 57790 is a novel and selective muscarinic M(2) receptor antagonist that releases acetylcholine and enhances cognition in experimental animals for the treatment of Alzheimer's disease. | |||
T7079 | Batefenterol | GSK961081,TD-5959 | Adrenergic Receptor , AChR |
Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor (Ki:1.4/1.3/3.7 nM). | |||
T8147 | Solifenacin | YM905 free base | AChR |
Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0, respectively. | |||
T0099 | Tolterodine tartrate | Detrol LA,PNU-200583E,Kabi-2234 | AChR |
Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo. |