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Search Results for " muscarinic receptor antagonist "

20

Compounds

Cat No. Product Name Synonyms Targets
T0218 Biperiden Bipariden,Akineton,KL 373,Biperidine AChR
Biperiden (Bipariden) is a muscarinic antagonist that has effects in both the central and peripheral nervous systems. It has been used in the treatment of arteriosclerotic, idiopathic, and postencephalitic parkinsonism. ...
T9771 Velufenacin AChR
Velufenacin is an antagonist of muscarinic receptor[1].
T23297 (S)-(+)-Dimethindene maleate AChR , Histamine Receptor
(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1, M3, and M4 receptors.
T16989 Tarafenacin D-tartrate SVT-40776 D-tartrate Others
Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.
T13992 CHF5407 SVT-47060 AChR
CHF5407(SVT-47060) is a potent and selective muscarinic M3 receptor antagonist with prolonged action at muscarinic receptors.CHF5407 has an effect on bronchospasm and may be used in the study of respiratory disorders.CHF...
T13385 Zamifenacin fumarate UK-76654 fumarate AChR
Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.
T6364 Desfesoterodine 5-HMT,(R)-5-Hydroxymethyl Tolterodine,PNU-200577,5-HM,5-hydroxymethyl Tolterodine AChR
Desfesoterodine (5-HMT) is a new muscarinic receptor antagonist with Kb of 0.84 nM.
T7895 Syn-Ake acetate Dipeptide diaminobutyroyl benzylamide AChR
Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.
T10914L Cyclodrine Cyclopent AChR
Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.
T10914 Cyclodrine hydrochloride AChR
Cyclodrine hydrochloride is a dual cholinergic muscarinic receptor (mAChR) and nicotinic receptor (nAChR) antagonist that can be used in the study of neurologically related diseases.
T1542 Pirenzepine dihydrochloride Pirenzepine HCl,Bisvanil,Tabe,LS519 AChR
Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.
T31207 GSK233705 Darotropium bromide,GSK 233705,GSK-233705B,GSK233705,GSK233705B,GSK-233705,GSK 233705B AChR
GSK233705 (Darotropium bromide) is a muscarinic receptor antagonist used in conjunction with the prevention and treatment of chronic obstructive pulmonary disease (COPD) and asthma in humans.
T5655 MAChR-IN-1 hydrochloride AChR
mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.
T23508 VU 0255035 AChR
muscarinic M1 antagonist
T29687 Afacifenacin Afacifenacin fumarate,SMP-986,NS 986,NS-986,SMP 986,NS986,SMP986 AChR
Afacifenacin (SMP-986) fumarate is an M3 muscarinic receptor-selective antagonist used in the study of ischemic heart disease, urinary incontinence and cystitis and other disorders.
T1534 Darifenacin hydrobromide Darifenacin HBr,UK-88525 AChR
Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and overactive bladder syndrome.
T28722 SCH 57790 SCH57790,SCH-57790 AChR
SCH 57790 is a novel and selective muscarinic M(2) receptor antagonist that releases acetylcholine and enhances cognition in experimental animals for the treatment of Alzheimer's disease.
T7079 Batefenterol GSK961081,TD-5959 Adrenergic Receptor , AChR
Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic and hβ2-adrenoceptor (Ki:1.4/1.3/3.7 nM).
T8147 Solifenacin YM905 free base AChR
Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0, respectively.
T0099 Tolterodine tartrate Detrol LA,PNU-200583E,Kabi-2234 AChR
Tolterodine tartrate (PNU-200583E) is a potent antagonist for muscarinic receptor. It show selectivity for the urinary bladder and salivary glands in vivo.
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TargetMol